Publication List

Original Papers;

78.Discovery, Characterization and Functional Improvement of Kumamonamide

as Novel Plant Growth Inhibitor that Disturb Plant Microtubules

T. Ishida*, H. Yoshimura, M. Takekawa, T. Higaki, T. Ideue, M. Hatano,

M. Igarashi, T. Tani, S. Sawa, H. Ishikawa*

Sci. Rep. DOI: 10.1038/s41598-021-85501-1

77. Epoxyquinophomopsins A and B from Endophytic Fungus Phomopsis sp.

and Their Activity against Tyrosine Kinase

E. Hermawati*, S. D. Ellita, L. D. Juliawaty, E. H. Hakim, Y. M. Syah, H. Ishikawa

J. Nat. Med. 75, 217–222 (2021).

76. Total Syntheses of (–)-Strictosidine and Related Indole Alkaloid Glycosides

J. Sakamoto, Y. Umeda, K. Rakumitsu, M. Sumimoto, H. Ishikawa*

Angew. Chem., Int. Ed. 59, 13414–13422 (2020).

75. 5,6-Dihydro-α-pyrones from the Leaves of Cryptocarya pulchinervia (Lauraceae)

L. D. Juliawaty*, P. N. Ra’idah, S. Abdurrahman, E. Hermawati, A. Alni,

M. I. Tan, H. Ishikawa, Y. M. Syah

J. Nat. Med. 74, 584–590 (2020).

74. Diaryliodonium Salt-Mediated Intramolecular C–N Bond Formation Using

Boron-Masking N-Hydroxyamides

M. Matsumoto, K. Wada, K. Urakawa, H. Ishikawa*

Org. Lett. 22, 781–785 (2020).

Selected “Cover Picture”. link

73.Identification of Naturally-Occurring Polyamines as Nematode Meloidogyne

incognita Attractants

M. Oota, A. Y.-L. Tsai, D. Aoki, Y. Matsushita, S. Toyoda, K. Fukushima,

K. Saeki, K. Toda, L. Perfus-Barbeoch, B. Favery, H. Ishikawa*, S. Sawa*

Mol. Plant 13, 658–665 (2020).

72. Enantioselective Total Synthesis of the Unnatural Enantiomer of Quinine

S. Shiomi, R. Misaka, M. Kaneko, H. Ishikawa*

Chem. Sci. 10, 9433–9437 (2019).

Selected “2019 Chemical Science HOT Article Collection” and

“Inside Front Cover”.

Highlighted in “Chemistry World” , “ChemistryViews”

and “Organic Chemistry Portal”

71. Total Syntheses of (–)-Secologanin, (–)-5-Carboxystrictosidine, and

　 (–)-Rubenine

K. Rakumitsu, J. Sakamoto, H. Ishikawa*

Chem. Eur. J., 25, 8996–9000 (2019).

　 Highlighted by Organic Chemistry Potal.

70.Enantioselective Construction of Octahydroquinolines via Trienamine-Mediated

Diels-Alder Reactions

T. Inoshita, K. Goshi, Y. Morinaga, Y. Umeda, H. Ishikawa*

Org. Lett., 21, 2903–2907 (2019).

69.Visualization of Plastid Peptidoglycan in the Charophyte Alga Klebsormidium

nitens Using a Metabolic Labeling Method

H. Takano*, T. Tsunefuka, S. Takio, H. Ishikawa, K. Takechi

Cytologia, 83, 375–380 (2018).

68.Two New Indolic and Quinolic Alkaloids and Other Secondary Metabolites from

Mostuea thomsonii (Loganiaceae)

E. G. B. Gompe, B. M. W. Ouahouo, V. T. Sielinou, M. Tsaffack, J. Fotie,

J. C. N. Assob, H. Ishikawa, P. Mkounga*, A. E. Nkengfack

Phytochemistry Letters, 26, 154–158 (2018).

67.α-Ketocarbenium Ions Derived from Orthoquinone-Containing Polycyclic Aromatic Compounds

K. Urakawa, Y. Kawabata, M. Mastuda, M. Sumimoto*, H. Ishikawa*

Org. Lett., 20, 2534–2537 (2018).

66. Total Syntheses and Stereochemical Reassignments of Mollenines A and B

S. Shiomi, K. Wada, Y. Umeda, H. Kato, S. Tsukamoto, H. Ishikawa*

Bioorg. Med. Chem. Lett. 28, 2766–2769 (2018).

Special issue “Prof. Dale L. Boger: A Celebration of 65 Years of Excellence”

65. Bioinspired Indole Prenylation Reaction in Water

S. Tanaka, S. Shiomi, H. Ishikawa*

J. Nat. Prod., 80, 2371–2378 (2017).

Selected “ACS Editors’ Choice” and “most accessed article in 2017 ranked 6th”.

64. Triterpenes and Coumaroyltyramide from Ochthocosmus Africanus

R. V. T. Sipowo, B. Marlyse, W. Ouahouo, H. L. D. Maza, H. Ishikawa,

H. Nishino, P. Mkounga*, A. E. Nkengfack

Journal of Diseases and Medicinal Plants, 3, 12–16 (2017).

63. Triterpenoids from Seeds of Tapinanthus Bangwensis

H. Maza, P. Mkounga*, S. L. Fenkam, S. K. Sado, H. Isikawa, H. Nishino,

E. A. Nkengfack

Phytochemistry Letters, 19, 23–29 (2017).

62.Acid–Mediated Aryl Migration Reaction of C–3 Aryl Substituted

Pyrrolidinoindolines

S. Tadano, H. Ishikawa*

Tetrahedron Lett., 58, 5–8 (2017).

61. New Lupan-type Triterpenoids

P. Mkounga*, H. L. D. Maza, B. M. W. Ouahouo, L. N. Tyon, H. Ishikawa,

H. Nishino, A. E. Nkengfack

Z. Naturforsch., 71, 381–386 (2016).

60. Moss Chloroplasts are Surrounded by a Peptidoglycan Wall Containing

D-Amino Acids

T.Hirano, K. Tanidokoro, Y. Shimizu, Y. Kawarabayashi, T. Ohshima, M. Sato,

S. Tadano, H. Ishikawa, S. Takio, K. Takechi, H. Takano*

The Plant Cell, 28,1521−1532 (2016).

　 Slelected “ Breakthrough report” and “Cover Picture”

59. Redox Switching of Orthoquinone-Containing Aromatic Compounds with

Hydrogen and Oxygen Gas

K. Urakawa, M. Sumimoto, M. Arisawa, M. Matsuda*, H. Ishikawa*

Angew. Chem., Int. Ed., 55, 7432–7436 (2016).

58. Collective Synthesis and Biological Evaluation of Tryptophan-based Dimeric

Diketopiperazine Alkaloids

S. Tadano, Y. Sugimachi, M. Sumimoto, S. Tsukamoto, H. Ishikawa*

Chem. Eur. J., 22, 1277–1291 (2016).

Selected “Hot Paper” and “Inside Cover Picture”

57. Efficient Organocatalytic Construction of C4-Alkyl Substituted Piperidines and

Their Application to the Synthesis of (+)-α-Skytanthine

S. Shiomi, E. Sugahara, H. Ishikawa*

Chem. Eur. J., 21, 14758–14763 (2015).

Highlighted by Organic Chemistry Portal

56. pH-driven, Reversible Epoxy Ring Opening/Closing in Graphene Oxide

T. Taniguchi, S. Kurihara, H. Tateishi, K. Hatakeyama, M. Konimura, H. Yokoi,

M. Hara, H. Ishikawa, Y. Matsumoto

Carbon 85, 560 (2015).

55. Organocatalyst-Mediated Dehydrogenation of Aldehydes to α, β-Unsaturated

Aldehydes, and Oxidative and Enantioselective Reaction of Aldehydes and

Nitromethane Catalyzed by Diphenylprolinol Silyl Ether

Y. Hayashi, T. Itoh, H. Ishikawa

Ads. Synth. Catal. 355, 3661 (2013).

54. One-Pot Synthesis of (–)-Oseltamivir and Mechanistic Insights

into the Organocatalyzed Michael Reaction

T. Mukaiyama, H. Ishikawa, H. Koshino, Y. Hayashi

Chem. Eur. J., 19, 17789 (2013).

53.Bio-Inspired Dimerization Reaction of Tryptophan Derivatives in Aqueous Acidic Media: Three-Step Syntheses of (+)-WIN 64821, (–)-Ditryptophenaline and (+)-Naseseazine B

S. Tadano, Y. Mukaeda, H. Ishikawa*

Angew. Chem., Int. Ed., 52, 7990 (2013).

52. Diarylprolinol in an Asymmetric Aldol Reaction of α-Alkyl-α-oxo Aldehyde as an

Electrophile

Y. Hayashi, Y. Yasui, M. Kojima, T. Kawamura, H. Ishikawa

Chem. Commun., 48, 4570 (2012).

51. Organocatalytic, Enantioselective Intramolecular [6+2] Cycloaddition

Reaction for the Formation of Tricyclopentanoids and Insight on Its Mechanism

from a Computational Study

Y. Hayashi, H. Gotoh, M. Honma, K. Sankar, I. Kumar, H. Ishikawa, K. Konno,

H. Yui, S. Tsuzuki, T. Uchimaru

J. Am. Chem. Soc., 113, 20175 (2011).

50. Spontaneous Conversion of 3-Alkyl-substituted 3-Hydroxyperoxypyrrolidine-2, 4-

diones into 5-Alkyl-5hydroxyoxazolidin-4-ones

M. A. Haque, H. Ishikawa, H. Nishino

Chem. Lett., 40, 1349 (2011).

49. Synthesis of (–)-Oseltamivir by Using a Microreactor in the Curtius

Rearrangement

H. Ishikawa, B. P. Bondzic, Y. Hayashi

Eur. J. Org. Chem., 6020 (2011).

48.One-pot Synthesis of Chiral Aziridines by a Domino Reaction using Desulfonylative Formation on the N-Tosyl Imine of Chloroacetaldehyde with an Asymmetric Mannich Reaction as a Key Step

Y.Hayashi, T. Urushima, D. Sakamoto, K. Torii, H. Ishikawa

Chem. Eur. J., 17, 11715 (2011).

47. Asymmetric Mannich Reaction of Imines Derived from Aliphatic and Aromatic

Aldehydes Catalyzed by Diarylprolinol Silyl Ether

T. Urushima, H. Ishikawa, Y. Hayashi

Chem. Eur. J., 17, 8273 (2011).

46. Organocatalyzed Michael Addition of Aldehyde to Nitro Alkenes – Generally

Accepted Mechanism Revisited and Revised

K. Patora-Komisarska, M. Benohoud, H. Ishikawa, D. Seebach, Y. Hayashi

Helv. Chim. Acta, 94, 719 (2011).

45. Oxidative and Enantioselective Cross-Coupling of Aldehydes and Nitromethane

Catalyzed by Diphenylprolinol Silyl Ether

Y. Hayashi, T. Itoh, H. Ishikawa,

Angew. Chem., Int. Ed., 50, 3920 (2011).

44.Asymmetric One-Pot Four-Component Coupling Reaction: Synthesis of Substituted Tetrahydropyranes Catalyzed by Diphenylprolinol Silyl Ether

H. Ishikawa, S. Sawano, Y. Yasui, Y. Shibata, Y. Hayashi

Angew. Chem., Int. Ed., 50, 3774 (2011).

43.One-Pot Synthesis of Chiral α-Substituted β,γ-Epoxy Aldehyde Derivatives through an Asymmetric Aldol Reaction of Chloroacetaldehyde

Y. Hayashi, Y. Yasui, T. Kawamura, M. Kojima, H. Ishikawa

Angew. Chem., Int. Ed., 50, 2804 (2011).

42.Diarylprolinol in the Direct Asymmetric Aldol Reaction of Trifluoromethylacetaldehyde Ethyl Hemiacetal with Aldehyde

Y. Hayashi, Y. Yasui, T. Kawamura, M. Kojima, H. Ishikawa

Synlett, 485 (2011).

41.One-Pot High-Yielding Synthesis of the DPP4-Selective Inhibitor ABT-341 by a Four Component Coupling Mediated by a Diphenylprolinol Silyl Ether

H. Ishikawa, M. Honma, Y. Hayashi

Angew. Chem., Int. Ed., 50, 2824 (2011).

Selected Very Important Paper and Inside Cover Picture

High lighted by Angew. Chem. Int. Ed. 50, 3605 (2011) and Nature Chemical

Biology 7, 190 (2011).

40.Asymmetric Epoxidation of α-Substituted Acroleins Catalyzed by Diphenylprolinol Silyl Ether

B. P. Bondzic, T. Urushima, H. Ishikawa, Y. Hayashi

Org. Lett., 12, 5434 (2010).

39.High-Yielding Synthesis of the Anti-Influenza Neuraminidase Inhibitor (−)-Oseltamivir by Two “One-Pot” Sequences

H. Ishikawa, T. Suzuki, H. Orita, T. Uchimaru, Y. Hayashi

Chem. Eur. J., 16, 12616 (2010).

38.Enantio- and Diastereoselective Synthesis of Piperidines by Coupling of Four Components in a “One-Pot” Sequence Involving Diphenylprolinol Silyl Ether Mediated Michael Reaction

T. Urushima, D. Sakamoto, H. Ishikawa, Y. Hayashi

Org. Lett., 12, 4588 (2010).

37.Polymeric Ethyl Glyoxylate in an Asymmetric Aldol Reaction Catalyzed by Diarylprolinol

T. Urushima, Y. Yasui, H. Ishikawa, Y. Hayashi

Org. Lett., 12, 2966 (2010).

36.One-Pot Synthesis of Chiral Bicyclo[3.3.0]octatrienes Using Diphenylprolinol Silyl Ether-Mediated Ene-Type Reaction

H. Gotoh, H. Ogino, H. Ishikawa, Y. Hayashi

Tetrahedron, 66, 4894 (2010).

35.Diphenylprolinol Silyl Ether as a Catalyst in an Asymmetric, Catalytic, and Direct Michael Reaction of Nitroethanol with α, β - Unsaturated Aldehydes

H. Gotoh, D. Okamura, H. Ishikawa, Y. Hayashi

Org. Lett., 11, 4056 (2009).

34.Asymmetric Aldol Reaction of Acetaldehyde and Isatin Derivatives for the Total Syntheses of ent-Convolutamydine E and CPC-1 and a Half Fragment of Madindoline A and B

T. Itoh, H. Ishikawa, Y. Hayashi

Org. Lett., 11, 3854 (2009).

33.Total Synthesis and Determination of The Absolute Configuration of FD-838, a Naturally Occurring Azaspirobicyclic Product

Y. Hayashi, K. Sankar, H. Ishikawa, Y. Nozawa, K. Mizoue, H. Kakeya

Bioorganic & Medicinal Chemistry Letters, 19, 3863 (2009).

32.Total Synthesis of Vinblastine, Vincristine, Related Natural Products, and Key Structural Analogues

H. Ishikawa, D. A. Colby, S. Seto, P. Va, A. Tam, H. Kakei, T. J. Rayl, I. Hwang,

D. L. Boger

J. Am. Chem. Soc., 131, 4904 (2009).

31.High-Yielding Synthesis of the Anti-Influenza Neuramidase Inhibitor (‐)-Oseltamivir by Three "One-Pot" Operations

H. Ishikawa, T. Suzuki, Y. Hayashi

Angew. Chem. Int. Ed., 48, 1304 (2009).

abstracted by Nature 457, 239 (2009).

30.Diphenylprolinol Silyl Ether as a Catalyst in an Enantioselective, Catalytic Michael Reaction for the Formation of α, α- Disubstituted α-Amino Acid Derivatives

Y. Hayashi, K. Obi, Y. Ohta, D. Okamura, H. Ishikawa

Chem. Asian. J., 4, 246 (2009).

29.Diphenylprolinol Silyl Ether Catalysis in an Asymmetric Formal Carbo [3 + 3] Cycloaddition Reaction via a Domino Michael/Knoevenagel Condensation

Y. Hayashi, M. Toyoshima, H. Gotoh, H. Ishikawa

Org. Lett., 11, 45 (2009).

28.Asymmetric, Catalytic, and Direct Self-Aldol Reaction of Acetaldehyde Catalyzed by Diarylprolinol

Y. Hayashi, S. Samanta, T. Itoh, H. Ishikawa

Org. Lett.,10, 5581, (2008).

27. Direct Organocatalytic Mannich Reaction of Acetaldehyde: An Improved Catalyst and Mechanistic Insight from a Computational Study

Y. Hayashi, T. Okano, T. Itoh, T. Urushima, H. Ishikawa, T. Uchimaru

Angew. Chem. Int. Ed., 47, 9053 (2008).

26.The Asymmetric Total Synthesis of (+)-Cytotrienin A, an Ansamycin-Type Anticancer Drug

Y. Hayashi, M. Shoji, H. Ishikawa, J. Yamaguchi, T. Tamura, H. Imai,

Y. Nishigaya, K. Takabe, H. Kakeya, H. Osada

Angew. Chem. Int. Ed., 47, 6657 (2008).

25.Asymmetric Diels-Alder Reactions of α, β -Unsaturated Aldehydes Catalyzed by a Diarylprolinol Silyl Ether Salt in the Presence of Water

Y. Hayashi, S. Samanta, H. Gotoh, H. Ishikawa

Angew. Chem. Int. Ed., 47, 6634 (2008).

24.The Effectiveness of Proteinogenic Amino Acids in theAsymmetric Aldol Reaction in DMSO and Aqueous DMSO

Y. Hayashi, T. Itoh, N. Nagae, M. Ohkubo, H. Ishikawa

Synlett, 2008,1565.

23.Asymmetric Michael Reaction of Acetaldehyde Catalyzed by Diphenylprolinol Silyl Ether

Y. Hayashi, T. Itoh, M. Ohkubo, H. Ishikawa

Angew. Chem. Int. Ed., 47, 4722 (2008).

22. Diphenylprolinol Silyl Ether as a Catalyst in an Enantioselective, Catalytic, Formal Aza [3+3] Cycloaddition Reaction for the Formation of Enantioenriched Piperidines

Y. Hayashi, H. Gotoh, R. Masui, H. Ishikawa

Angew. Chem. Int. Ed., 47, 4012 (2008).

21.Proline-Mediated Enantioselective Construction of Tetrahydropyrans via a Domino Aldol/Acetalization Reaction

D. Hazelard, H. Ishikawa, D. Hashizume, H. Koshino, Y. Hayashi

Org. Lett., 10, 1445 (2008).

20.A Diarylprolinol in an Asymmetric, Catalytic, and Direct Crossed-Aldol Reaction of Acetaldehyde

Y. Hayashi, T. Itoh, S. Aratake, H. Ishikawa

Angew. Chem. Int. Ed., 47, 2082 (2008).

19.Direct Coupling of Catharanthine and Vindoline to Provide Vinblastine: Total Synthesis of (+)- and ent-(-)-Vinblastine

H. Ishikawa, D. A. Colby, D. L. Boger

J. Am. Chem. Soc., 130, 420 (2008).

18.Diphenylprolinol Silyl Ether as Catalyst of an Asymmetric, Catalytic, and Direct Michael Reaction of Nitroalkanes with α,β -Unsaturated Aldehydes

H. Gotoh, H. Ishikawa, Y. Hayashi

Org. Lett., 9, 5307 (2007).

17.Total Synthesis of (-)- and ent-(+)-4-Desacetoxy-5-desethylvindoline

H. Ishikawa and Dale L. Boger

Heterocycles, 72, 95 (2007).

Commemorative issue honoring Professor Y. Kishi on his 70th birthday.

16.New Procedure to Mask the 2,3-π Bond of the Indole Nucleus and Its Application to the Preparation of Potent Opioid Receptor Agonists with a Corynanthe Skeleton

H. Takayama, K. Misawa, N. Okada, H. Ishikawa, M. Kitajima, Y. Hatori,

T. Murayama, S. Wongseripipatana, K. Tashima, K. Matsumoto, S. Horie

Org. Lett., 8, 5705 (2006).

15.Total Synthesis of (-)- and ent-(+)-Vindoline and Related Alkaloids

H. Ishikawa, G. I. Elliott, J. Velcicky, Y. Choi, D. L. Boger

J. Am. Chem. Soc., 128, 10596 (2006).

14.Intramolecular Diels-Alder/1,3-Dipolar Cycloaddition Cascade of 1,3,4-Oxadiazoles

G. I. Elliott, J. R. Fuchs, B. S. J. Blagg, H. Ishikawa, H. Tao, Z. Yuan,

D. L. Boger

J. Am. Chem. Soc., 128, 10589 (2006).

13.Partial Agonistic Effect of 9-Hydroxycorynantheidine on μ-Opioid Receptor in The Guinea- Pig Ileum

K. Matsumoto, H. Takayama, H. Ishikawa, N. Aimi, D. Ponglux, K. Watanabe,

S. Horie

Life Sciences, 78, 2265 (2006).

12.Total Synthesis of (-)- and ent-(+)-Vindorosine; Tandem Intramolecular Diels-Alder/1,3-Dipolar Cycloaddition of 1,3,4-Oxadiazoles

G. I. Elliott, J. Velcicky, H. Ishikawa, Y. Li, D. L. Boger

Angew. Chem., Int. Ed., 45, 620 (2006).

selected Very Important Paper

11.Total Synthesis of Natural-(-)- and ent-(+)-Vindoline

Y. Choi, H. Ishikawa, J. Velcicky, G. I. Elliott, M. M. Miller, D. L. Boger

Org. Lett., 7, 4539 (2005).

10.Total Synthesis of Natural (+)- and ent-(-)-4-Desacetoxy-6,7-dihydrovindorosine and Natural and ent-Minovine: Oxadiazole Tandem Intramolecular Diels-Alder/1,3-Dipolar Cycloaddition Reaction

Z. Yuan, H. Ishikawa, D. L. Boger

Org. Lett., 7, 737 (2005).

9.Antinociception, Tolerance and Withdrawal Symptoms Induced by 7-Hydroxymitragynine, an Alkaloid from The Thai Medicinal Herb Mitragyna speciosa

K. Matsumoto, S. Horie, H. Takayama, H. Ishikawa, N. Aimi, D. Ponglux,

T. Murayama, K. Watanabe

Life Sciences, 78, 2 (2005).

8.Indole Alkaloids of a Thai Medicinal Herb, Mitragyna speciosa, that has Opioid Agonistic Effect in Guinea-pig Ileum

S. Horie, F. Koyama, H. Takayama, H. Ishikawa, N.Aimi, D. Ponglux,

K. Matsumoto,T. Murayama

Planta Med., 71, 231 (2005).

7.m-Chloroperbenzoic Acid Oxidation of Corynanthe-type Indole Alkaloid, Mitragynine, Afforded Unusual Dimerization Products

H. Ishikawa, M. Kitajima, H. Takayama

Heterocycles, 63, 2597 (2004).

6.Antinociceptive Effect of 7-Hydroxymitragynine in Mice: Discovery of an Orally Active Opioid Analgesic from the Thai Medical Herb Mitragyna speciosa

K. Matsumoto, S. Horie, H. Ishikawa, H. Takayama, N. Aimi, D. Ponglux,

K. Watanabe

Life Sciences, 74, 2143 (2004).

5.A New 9-Methoxyyohimbine type Indole Alkaloid from Mitragyna africanus

H. Takayama, H. Ishikawa, M. Kitajima, N. Aimi, B. M. Aji

Chem. Pharm. Bull., 52, 359 (2004).

4.Dimerization of Indole Derivatives with Hypervalent Iodines (III): a New Entry for the Concise Total Synthesis of rac- and meso-Chimonanthines

H. Ishikawa, H. Takayama, N. Aimi

Tetrahedron Lett., 43, 5637 (2002).

3.Formation of an Unusual Dimeric Compound by Lead Tetraacetate Oxidation of a Corynanthe-Type Indole Alkaloid, Mitragynine

H. Takayama, H. Ishikawa, M. Kitajima, N. Aimi

Chem. Pharm. Bull., 50, 960 (2002).

2.Studies on the Synthesis and Opioid Agonistic Activities of Mitragynine-Related Indole Alkaloids: Discovery of Opioid Agonists Structurally Different from Other Opioid Ligands

H. Takayama, H. Ishikawa, M. Kurihara, M. Kitajima, N. Aimi, D. Ponglux,

F. Koyama, K. Matsumoto, T. Moriyama, L. T. Yamatomo, K. Watanabe,

T. Murayama, S. Horie

J. Med. Chem., 45, 1949 (2002).

1.Structure Revision of Mitragynaline, an Indole Alkaloid in Mitragyna speciosa

H. Takayama, H. Ishikawa, M. Kurihara, M. Kitajima, S. Sakai, N. Aimi, H. Seki,

K. Yamaguchi, I. M. Said, P. J. Houghton

Tetrahedron Lett., 42, 1741 (2001).

Review;

9.非天然型キニーネの実用的全合成を目指して

石川勇人

　有機合成化学協会誌（J. Syn. Org. Chem. Jpn.）, 76, 414－417 (2018).

8. Unified Total Synthesis of Tryptophan-based Dimeric Diketopiperazine Alkaloids

H. Ishikawa*

有機合成化学協会誌（J. Syn. Org. Chem. Jpn.）, 74, 104–116 (2016).

(Invited review article for Incentive Award in Synthetic Organic Chemistry, Japan)

7.　Alkaloid Synthesis using Chiral Secondary Amine Organocatalysts

H. Ishikawa*, S. Shiomi

Org. Biomol. Chem., 14, 409-424 (2016); DOI: 10.1039/C5OB02021B

6. 生物に倣うインドール酸化反応を用いた生物活性アルカロイドの全合成

　　石川勇人

　　YAKUGAKU ZASSHI, 135, 383–390 (2015).

5.　ポットエコノミーを指向した効率的天然物合成

　石川勇人、林雄二郎

　ファインケミカル（特集号　天然物合成化学の新たな展開），43, 6 (2014).

4.　Synthesis of Tryptophan-based Dimeric Diketopiperazine Alkaloids using

Bio-inspired Reactions

S.Tadano, H. Ishikawa*

Synlett, 25, 157-162 (2014). (Invaited Article as Synpacts: review article)

3. 有機触媒を用いた（−）‐オセルタミビルの３ポット合成

石川勇人、林雄二郎

ファインケミカル（特集号　創意工夫が導く高度ワンポット合成）,

　　 39, 5 (2010).

2. インフルエンザ治療薬オセルタミビルの３ポット合成―ジフェニルプロリノール

シリルエーテル触媒を用いた全合成―

石川勇人、林雄二郎

化学と生物, 48, 156 (2010).

1. Total Synthesis of Vindoline and Related Alkaloids

　　H. Ishikawa, D. L. Boger

有機合成化学協会誌（J. Syn. Org. Chem. Jpn.）, 67, 123 (2009).

Books;

6. The Alkaloids, Elsevier, Vol 79, 2018

Alkaloid Synthesis using Organocatalyst

Hayato Ishikawa*, Shinya Shiomi, pp. 1–70.

5. 天然物の全合成　（CSJカレントレビュー29）化学同人、2018

Chap. 5「生合成を参考にした全合成」pp78–85.

および basic concept 「連続反応の基礎」 pp 30–35.

　石川勇人

4. 有機分子触媒の開発と工業利用（監修　秋山隆彦）、CMC出版、2018

　第27章二級アミン型不斉有機触媒反応の実用化に向けた触媒量低減化と

　アルカロイド合成への応用、pp 295–304.

　石川勇人

3. アルカロイドの科学（監修　高山廣光）、化学同人、2017

　第14章　有機触媒を利用したアルカロイドの不斉合成、 pp.283–300

　石川勇人

2. 有機分子触媒の化学　（CSJカレントレビュー22）化学同人、2016

　 Chap. 18、有用物質（医薬品等）への応用、 pp.195–201.

　林雄二郎、石川勇人

1. Asymmetric Synthesis II: More Methods and Applications; Edited by Mathias

Christmann, Stefan Brase, WILEY-VCH, 2013

Chap. 9, Total Synthesis of Oseltamivir and ABT-341 Using One-Pot Technology,

Hayato Ishikawa and Yujiro Hayashi, pp 61.

Invited Articles and Others;

3. 熊本におけるアイラトビカズラ（マメ科）のDNAシーケンスによる種同定

　岡本竜弥、相田光宏、石川勇人、澤進一郎

　 BOTANY 70号（熊本記念植物採集会）、pp. 8－10、2020年.

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